SCD1 inhibitor-4

CAS No. 1295541-87-5

SCD1 inhibitor-4( —— )

Catalog No. M23453 CAS No. 1295541-87-5

SCD1 inhibitor-4 is stearoylCoA desaturase-1 (SCD1) inhibitor. SCD1 inhibitor-4 can be used for the research of diabetes.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 58 In Stock
5MG 87 In Stock
10MG 158 In Stock
25MG 320 In Stock
50MG 515 In Stock
100MG 740 In Stock
500MG 1521 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    SCD1 inhibitor-4
  • Note
    Research use only, not for human use.
  • Brief Description
    SCD1 inhibitor-4 is stearoylCoA desaturase-1 (SCD1) inhibitor. SCD1 inhibitor-4 can be used for the research of diabetes.
  • Description
    SCD1 inhibitor-4 is stearoylCoA desaturase-1 (SCD1) inhibitor. SCD1 inhibitor-4 can be used for the research of diabetes.
  • In Vitro
    ——
  • In Vivo
    SCD1 inhibitor-4 (1~30 mg/kg) shows a dose-dependent decrease in desaturation index with a 55 % reduction at 1 mg/kg and 85% reduction at the 10 and 30 mg/kg doses.
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Dehydrogenase
  • Recptor
    SCD1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1295541-87-5
  • Formula Weight
    363.34
  • Molecular Formula
    C17H16F3N5O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 90 mg/mL?(247.70 mM;?Need ultrasonic)
  • SMILES
    O=C(C1=C(C)N(CC2=CC=CC(C(F)(F)F)=C2)C=N1)NC3=NN(C)C=C3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Atkinson KA, et al. N-benzylimidazole carboxamides as potent, orally active stearoylCoA desaturase-1 inhibitors. Bioorg Med Chem Lett. 2011;21(6):1621-1625.
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